SCHEMBL8380299

SCHEMBL8380299

CC/C=C/[C@H]1CC[C@H](c2cnc(-c3ccc(F)c(F)c3)nc2)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.34
NPY5R Q15761 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
GRIN2B Q13224 8/20 0.32
RXRA P19793 6/20 0.32
GRIN1 Q05586 6/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
DHODH Q02127 2/20 0.31
PDE5A O76074 1/20 0.31
HDAC4 P56524 1/20 0.31
GRM2 Q14416 1/20 0.31
USP7 Q93009 1/20 0.31
OPRL1 P41146 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9312803 1.00 ACACB (0.34) ACACBNPY5RCYP11B1CYP11B2GRIN2B
SCHEMBL8382535 0.91 ACACB (0.35) ACACBNPY5RCYP11B1CYP11B2GRIN2B
SCHEMBL8382537 0.91 ACACB (0.35) ACACBNPY5RCYP11B1CYP11B2GRIN2B
SCHEMBL9311907 0.91 ACACB (0.35) ACACBNPY5RCYP11B1CYP11B2GRIN2B
SCHEMBL8383724 0.90 CYP11B1 (0.36) ACACBCYP11B1CYP11B2GRIN2BRXRA
SCHEMBL9312474 0.90 CHRNB1 (0.35) CYP11B1CYP11B2GRIN2BGRIN1DHODH
SCHEMBL8380287 0.90 CHRNB1 (0.35) CYP11B1CYP11B2GRIN2BGRIN1DHODH
SCHEMBL9313556 0.90 CYP11B1 (0.36) ACACBCYP11B1CYP11B2GRIN2BRXRA
SCHEMBL8380279 0.87 KDM1A (0.40) CYP11B1CYP11B2GRM2ALDH1A1CYP1A2
SCHEMBL9312015 0.87 KDM1A (0.40) CYP11B1CYP11B2GRM2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475273-B1 Liquid crystal mixture containing halogenated alcenyl compounds MERCK PATENT GMBH (DE) 1999-04-07 EP disclosed
US-5292452-A Electrooptical devices; high dielectric anisotropy, low rotation viscosity, short response time HOFFMANN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0475273-A1 Halogenated alcenyl compounds F. HOFFMANN-LA ROCHE AG (CH) 1992-03-18 EP disclosed