SCHEMBL8380931

SCHEMBL8380931

COC(=O)C=Cc1ccc(OCCC(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.51
KMT2A Q03164 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
KDM1A O60341 1/20 0.51
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
TYR P14679 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
GSK3B P49841 1/20 0.48
BACE1 P56817 1/20 0.48
MAPT P10636 3/20 0.47
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
FDPS P14324 1/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8380930 1.00 PPARA (0.51) PPARAKMT2ASMN1; SMN2KDM1ACA12
SCHEMBL8381015 0.87 PPARA (0.52) PPARAKMT2ASMN1; SMN2GSK3BBACE1
SCHEMBL8381018 0.87 PPARA (0.52) PPARAKMT2ASMN1; SMN2GSK3BBACE1
SCHEMBL5207328 0.85 PPARA (0.58) PPARAKMT2ASMN1; SMN2KDM1ACA12
SCHEMBL8380557 0.81 SMN1; SMN2 (0.62) KMT2ASMN1; SMN2MAPTRAB9AALDH1A1
SCHEMBL8213995 0.81 AKR1B10 (0.61) PPARAKMT2ASMN1; SMN2GSK3BBACE1
SCHEMBL8782823 0.79 ABCG2 (0.62) PPARASMN1; SMN2CA12CA1CA2
SCHEMBL13958437 0.79 CA12 (0.58) PPARAKMT2ASMN1; SMN2CA12CA1
SCHEMBL142092 0.79 ABCG2 (0.62) PPARASMN1; SMN2CA12CA1CA2
SCHEMBL19244469 0.79 ABCG2 (0.62) KMT2ACA12CA1CA2TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874436-A EFFECTIVE IN INHIBITING THE ACTION OF A BACTERIAL HISTIDINE PROTEIN KINASE; USEFUL AGAINST ANTIBIOTIC RESISTANT ORGANISMS DEMERS JAMES P (US) 1999-02-23 US disclosed
WO-1997048676-A1 TRIPHENYLALKYL ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-12-24 WO disclosed
US-5643950-A INHIBITORS OF A BACTERIAL HISTIDINE PROTEIN KINASE ORTHO PHARMACEUTICAL CORPORATION (US) 1997-07-01 US disclosed