SCHEMBL8383166

SCHEMBL8383166

O=C(Nc1ccc2sccc2c1)c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.56
RAB9A P51151 8/20 0.56
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
TP53 P04637 2/20 0.56
NFKB1 P19838 2/20 0.56
NFKB2 Q00653 2/20 0.56
RELA Q04206 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
NAMPT P43490 1/20 0.54
GAA P10253 1/20 0.54
PTPN1 P18031 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
MITF O75030 1/20 0.53
KCNK3 O14649 1/20 0.52
KCNK9 Q9NPC2 1/20 0.52
ESR1 P03372 1/20 0.52
SNCA P37840 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4251091 0.80 GAA (0.61) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL10116570 0.78 HDAC8 (0.50) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL10114494 0.78 HDAC8 (0.50) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL14424314 0.77 HDAC8 (0.49) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL2304786 0.77 NPC1 (0.54) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL4315507 0.77 MEN1 (0.58) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL13201004 0.77 NAMPT (0.71) NPC1RAB9AMEN1KMT2ANFKB1
SCHEMBL10684470 0.76 PTPN1 (0.88) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL30093465 0.75 NPC1 (0.57) NPC1RAB9AMEN1KMT2ATP53
SCHEMBL8385383 0.75 MEN1 (0.54) NPC1RAB9AMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874427-A MIGRAINE ELI LILLY AND COMPANY (US) 1999-02-23 US disclosed
EP-0875513-A1 Substituted heteroaromatic 5-HT 1F agonists ELI LILLY AND COMPANY (US) 1998-11-04 EP disclosed
WO-1998046570-A1 SUBSTITUTED HETEROAROMATIC 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed