SCHEMBL8387409

SCHEMBL8387409

Cc1c(-c2cc(F)cc(C(F)(F)F)c2)ccc(N)c1C#N

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
PGR P06401 1/20 0.34
PTGS1 P23219 1/20 0.33
NLRP3 Q96P20 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
HTT P42858 2/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
NCOA1 Q15788 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HIF1A Q16665 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
DHODH Q02127 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8386061 0.92 CTSS (0.37) RXRARXRBNLRP3ALOX5APFEN1
SCHEMBL8651015 0.80 ABL1 (0.35) PTGS1ALOX5APFEN1HTTALDH1A1
SCHEMBL8387382 0.75 AKR1C3 (0.36) NLRP3ALOX5APFEN1HTTCTSS
SCHEMBL23915997 0.74 ALOX5AP (0.44) RXRARXRBRXRGALOX5APFEN1
SCHEMBL8387020 0.73 KDM4E (0.42) HTTLMNAPOLBHIF1AALDH1A1
SCHEMBL8388339 0.72 IKBKB (0.42) HTTCTSSCTSKLMNAPOLB
SCHEMBL8390382 0.72 ADORA2A (0.44) HTTSMN1; SMN2ALDH1A1MAPTPKM
SCHEMBL8649829 0.70 IKBKB (0.40) ALOX5APFEN1HTTCTSSCTSK
SCHEMBL8390378 0.69 MAOB (0.32)
SCHEMBL8385922 0.68 DHFR (0.39) PTGS1ALDH1A1MAPTHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874579-A Insecticidal substituted-2.4-diaminoquinazolines related applications FMC CORPORATION (US) 1999-02-23 US disclosed
US-5616718-A USEFUL FOR MAKING 2,4-DIAMINOQUINAZOLINES; INSECTICIDES FMC CORPORATION (US) 1997-04-01 US disclosed
US-5534518-A Insecticidal substituted-2,4-diaminoquinazolines FMC CORPORATION (US) 1996-07-09 US disclosed
EP-0684824-A4 INSECTICIDAL SUBSTITUTED-2,4-DIAMINOQUINAZOLINES. FMC CORP (US) 1996-02-14 EP disclosed
EP-0684824-A1 INSECTICIDAL SUBSTITUTED-2,4-DIAMINOQUINAZOLINES FMC CORPORATION (US) 1995-12-06 EP disclosed
WO-1994018980-A1 INSECTICIDAL SUBSTITUTED-2,4-DIAMINOQUINAZOLINES FMC CORPORATION (US) 1994-09-01 WO disclosed