SCHEMBL8394170

SCHEMBL8394170

O=S(=O)(Nc1ccc(Cl)nc1)c1cccc2ccccc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 4/20 0.67
TSHR P16473 2/20 0.56
PGR P06401 1/20 0.56
RORA P35398 1/20 0.51
RORC P51449 1/20 0.51
NR1H2 P55055 1/20 0.51
NR1H4 Q96RI1 1/20 0.51
ALDH1A1 P00352 2/20 0.50
HTT P42858 2/20 0.50
NR1I2 O75469 1/20 0.50
PFKFB3 Q16875 1/20 0.50
CYP17A1 P05093 1/20 0.49
HDAC1 Q13547 1/20 0.49
SGK1 O00141 1/20 0.48
PTPN2 P17706 1/20 0.48
PTPN1 P18031 1/20 0.48
PTPN5 P54829 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HCRTR1 O43613 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8392200 0.83 EDNRA (0.67) EDNRATSHRPGRRORARORC
SCHEMBL8055281 0.81 EDNRA (1.00) EDNRA
SCHEMBL8394279 0.81 EDNRA (0.67) EDNRATSHRPGRALDH1A1MEN1
SCHEMBL27415009 0.80 P4HTM (0.67) TSHRPGRRORARORCNR1H2
SCHEMBL8392321 0.80 EDNRA (0.66) EDNRATSHRPGRRORARORC
SCHEMBL6409546 0.78 TSHR (0.67) TSHRPGRRORARORCNR1H2
SCHEMBL8390387 0.77 EDNRA (0.66) EDNRATSHRPGRRORARORC
SCHEMBL9140469 0.77 TSHR (0.55) EDNRATSHRPGRRORARORC
SCHEMBL812673 0.77 TSHR (0.74) EDNRATSHRPGRRORARORC
SCHEMBL31110643 0.77 TSHR (0.74) EDNRATSHRPGRRORARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752986-B1 N-HETEROCYCLYL SULPHONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LTD (GB) 1999-05-19 EP disclosed