SCHEMBL8396249

SCHEMBL8396249

COc1ccccc1N(Cc1nc2ccc(F)c(F)c2s1)C(=O)CCC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
TSPO P30536 3/20 0.38
KDM4E B2RXH2 3/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
HSD17B10 Q99714 3/20 0.36
TSHR P16473 2/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8400564 0.90 ALDH1A1 (0.39) ALDH1A1TSPOKDM4EKMT2APOLB
SCHEMBL8395613 0.88 AKR1B1 (0.36) ALDH1A1KMT2APOLBTDP1TSHR
SCHEMBL8395480 0.87 AKR1B1 (0.40) KMT2APOLBTSHR
SCHEMBL8398844 0.86 AKR1B1 (0.42) ALDH1A1TSPOKDM4EKMT2APOLB
SCHEMBL8518212 0.85 AKR1B1 (0.34)
SCHEMBL8396414 0.85 AKR1B1 (0.36) KMT2APOLBTSHR
SCHEMBL8399154 0.85 AKR1B1 (0.35) ALDH1A1KDM4EKMT2APOLBTSHR
SCHEMBL8396110 0.85 AKR1B1 (0.41) ALDH1A1TSPOKDM4EKMT2ATDP1
SCHEMBL8399078 0.84 AKR1B1 (0.46)
SCHEMBL8395274 0.84 AKR1B1 (0.37) ALDH1A1POLBTSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed