SCHEMBL8395274

SCHEMBL8395274

O=C(O)CCC(=O)N(Cc1nc2ccc(F)c(F)c2s1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.37
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
HTT P42858 2/20 0.35
ALOX15 P16050 1/20 0.35
AKR1A1 P14550 2/20 0.35
NAAA Q02083 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
TSHR P16473 1/20 0.34
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
RAB9A P51151 1/20 0.33
PAX8 Q06710 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8400228 0.92 LTB4R2 (0.35) AKR1B1TP53TSHRALDH1A1
SCHEMBL8399344 0.91 HDAC6 (0.37) AKR1B1AKR1A1TP53
SCHEMBL8399085 0.91 LTB4R2 (0.40) TP53NPC1
SCHEMBL8399247 0.90 AKR1B1 (0.32) AKR1B1AKR1A1
SCHEMBL8399708 0.90 AKR1B1 (0.35) AKR1B1SMN1; SMN2TP53
SCHEMBL8399483 0.90 HDAC6 (0.39) SMN1; SMN2HTTNPC1ALDH1A1RAB9A
SCHEMBL8395613 0.89 AKR1B1 (0.36) AKR1B1SMN1; SMN2HTTALOX15AKR1A1
SCHEMBL8398137 0.89 RAB9A (0.40) AKR1B1HTTTP53POLBNPC1
SCHEMBL8396627 0.89 RXRA (0.34) AKR1B1SMN1; SMN2HTTAKR1A1
SCHEMBL8399251 0.88 TSHR (0.40) AKR1B1HPGDAKR1A1TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed