SCHEMBL8396288

SCHEMBL8396288

CSc1cccc(N(Cc2nc3c(Cl)c(Cl)ccc3s2)C(=O)CCC(=O)O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.38
HDAC6 Q9UBN7 2/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32
GRIN3A Q8TCU5 2/20 0.32
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32
NPC1 O15118 1/20 0.32
JAK2 O60674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8395876 0.91 AKR1B1 (0.37) AKR1B1HDAC6MEN1KMT2ANPC1
SCHEMBL8399715 0.90 SMN1; SMN2 (0.39) AKR1B1HDAC6MEN1KMT2AGRIN2D
SCHEMBL8400332 0.89 RAB9A (0.43) AKR1B1HDAC6MEN1KMT2AMAPT
SCHEMBL8397937 0.89 AKR1B1 (0.38) AKR1B1HDAC6MEN1KMT2AMAPT
SCHEMBL8400428 0.88 AKR1B1 (0.41) AKR1B1HDAC6MEN1KMT2AMAPT
SCHEMBL8398067 0.86 AKR1B1 (0.46) AKR1B1HDAC6MEN1KMT2AMAPT
SCHEMBL8395578 0.86 AKR1B1 (0.39) AKR1B1HDAC6MEN1KMT2AMAPT
SCHEMBL8396282 0.86 AKR1B1 (0.40) AKR1B1HDAC6MEN1KMT2ANPC1
SCHEMBL8397855 0.86 AKR1B1 (0.40) AKR1B1HDAC6MEN1KMT2AMAPT
SCHEMBL8399147 0.85 MTNR1A (0.39) AKR1B1KMT2AMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed