SCHEMBL8397923

SCHEMBL8397923

Cc1cccc(N(Cc2nc3cc(F)cc(F)c3s2)C(=O)CCC(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 6/20 0.42
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
JAK2 O60674 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
PAX8 Q06710 1/20 0.40
TP53 P04637 2/20 0.38
LMNA P02545 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
LTB4R2 Q9NPC1 2/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.37
THRB P10828 1/20 0.37
F2 P00734 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399118 0.91 AKR1B1 (0.43) AKR1B1NPC1LTB4R2KMT2AMEN1
SCHEMBL8397936 0.90 AKR1B1 (0.48) AKR1B1LMNA
SCHEMBL8399130 0.90 SMN1; SMN2 (0.41) AKR1B1RAB9ANPC1JAK2ALDH1A1
SCHEMBL8399244 0.89 AKR1B1 (0.44) AKR1B1KMT2AMEN1
SCHEMBL8399158 0.89 AKR1B1 (0.41) AKR1B1LMNALTB4R2
SCHEMBL8398031 0.89 AKR1B1 (0.42) AKR1B1LMNALTB4R2KMT2A
SCHEMBL8396406 0.89 AKR1B1 (0.46) AKR1B1RAB9ANPC1ALDH1A1HTT
SCHEMBL8398694 0.88 AKR1B1 (0.40) AKR1B1LMNALTB4R2
SCHEMBL8398176 0.88 AKR1B1 (0.40) AKR1B1LTB4R2KMT2AMEN1F2
SCHEMBL8396078 0.87 LTB4R2 (0.40) AKR1B1TP53LMNALTB4R2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed