SCHEMBL8397971

SCHEMBL8397971

CCOC(=O)[C@H](OS(=O)(=O)C(F)(F)F)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
MAPT P10636 2/20 0.34
HSD17B10 Q99714 2/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PIN1 Q13526 1/20 0.33
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
ALDH1A1 P00352 4/20 0.31
LMNA P02545 1/20 0.30
ATM Q13315 1/20 0.30
CXCR2 P25025 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP3 P08254 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8397975 1.00 POLB (0.36) POLBMAPTHSD17B10HTTSMN1; SMN2
SCHEMBL1576184 0.82 CA14 (0.40) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL701746 0.82 POLB (0.38) POLBMAPTHSD17B10HTTSMN1; SMN2
SCHEMBL324715 0.82 POLB (0.38) POLBMAPTHSD17B10HTTSMN1; SMN2
SCHEMBL324716 0.82 POLB (0.38) POLBMAPTHSD17B10HTTSMN1; SMN2
SCHEMBL8400666 0.80 MMP1 (0.38) CA1CA2CXCR2MMP1MMP2
SCHEMBL29205828 0.80 MMP1 (0.38) CA1CA2CXCR2MMP1MMP2
SCHEMBL9773131 0.79 MMP8 (0.43) POLBMAPTHSD17B10HTTSMN1; SMN2
SCHEMBL31153798 0.79 CA12 (0.34) CA12CA1CA2CXCR2
SCHEMBL5551942 0.79 CA12 (0.34) CA12CA1CA2CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918757-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1999-06-02 EP disclosed
WO-1997043268-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1997-11-20 WO disclosed