SCHEMBL8399188

SCHEMBL8399188

COc1ccc(NC(N)=O)cc1N1CCN(C)CC1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 19/20 0.67
HTR1B P28222 17/20 0.67
HTR1A P08908 16/20 0.67
HTR2C P28335 8/20 0.67
HTR2A P28223 8/20 0.67
HTR6 P50406 6/20 0.67
HTR7 P34969 2/20 0.67
TMPRSS2 O15393 1/20 0.59
SLC6A4 P31645 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22411115 0.83 HTR1A (0.79) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8402123 0.83 HTR1D (0.65) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL14734295 0.82 HTR1D (0.62) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8759779 0.81 HTR1A (1.00) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8704883 0.81 HTR1D (0.70) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL7525124 0.81 HTR1D (0.66) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8122186 0.81 MEN1 (0.60) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8705195 0.81 HTR1D (0.70) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8705402 0.81 HTR1D (0.70) HTR1DHTR1BHTR1AHTR2CHTR2A
SCHEMBL8663635 0.81 HTR1A (0.76) HTR1DHTR1BHTR1AHTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5905080-A Amide and urea derivatives as 5HT1D receptor antagonists SMITHKLINE BEECHAM, P.L.C. (GB) 1999-05-18 US claimed
WO-2020183011-A1 HTR1D INHIBITORS AND USES THEREOF IN THE TREATMENT OF CANCER INSTITUT CURIE (FR) 2020-09-17 WO disclosed
US-5905080-A Amide and urea derivatives as 5HT1D receptor antagonists SMITHKLINE BEECHAM, P.L.C. (GB) 1999-05-18 US disclosed