SCHEMBL8399278

SCHEMBL8399278

COc1ccccc1N(Cc1nc2c(Cl)c(Cl)ccc2s1)C(=O)CCC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.41
ALDH1A1 P00352 7/20 0.38
KDM4E B2RXH2 4/20 0.38
HSD17B10 Q99714 4/20 0.37
POLB P06746 3/20 0.37
USP5 P45974 1/20 0.37
BRAP Q7Z569 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
USP16 Q9Y5T5 1/20 0.37
USP3 Q9Y6I4 1/20 0.37
TSHR P16473 3/20 0.36
GAA P10253 2/20 0.36
CCR6 P51684 1/20 0.36
PAX8 Q06710 1/20 0.36
KMT2A Q03164 3/20 0.36
STING1 Q86WV6 3/20 0.36
MEN1 O00255 2/20 0.36
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399110 0.90 ALDH1A1 (0.39) AKR1B1ALDH1A1KDM4EHSD17B10POLB
SCHEMBL8396244 0.88 AKR1B1 (0.45) AKR1B1ALDH1A1KDM4EPOLBHDAC6
SCHEMBL8400221 0.87 AKR1B1 (0.43) AKR1B1POLBHDAC6GAAPAX8
SCHEMBL8399303 0.85 AKR1B1 (0.43) AKR1B1POLBHDAC6TSHRGAA
SCHEMBL8398174 0.85 AKR1B1 (0.43) AKR1B1ALDH1A1POLBHDAC6GAA
SCHEMBL8396110 0.85 AKR1B1 (0.41) AKR1B1ALDH1A1KDM4EHSD17B10TSHR
SCHEMBL8400252 0.85 AKR1B1 (0.41) AKR1B1ALDH1A1POLBHDAC6TSHR
SCHEMBL8398067 0.84 AKR1B1 (0.46) AKR1B1ALDH1A1POLBHDAC6TSHR
SCHEMBL8396279 0.83 USP2 (0.40) AKR1B1ALDH1A1POLBTSHRGAA
SCHEMBL8399147 0.81 MTNR1A (0.39) AKR1B1KMT2ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed