SCHEMBL8400418

SCHEMBL8400418

Cc1cccc(N(Cc2nc3c(F)c(F)ccc3s2)C(=O)CCC(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
JAK2 O60674 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
PAX8 Q06710 1/20 0.40
AKR1B1 P15121 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
POLQ O75417 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399142 0.90 AKR1B1 (0.41) NPC1AKR1B1LTB4R2KMT2AMEN1
SCHEMBL8395834 0.90 SMN1; SMN2 (0.41) RAB9ANPC1JAK2ALDH1A1HTT
SCHEMBL8518906 0.89 AKR1B1 (0.40) AKR1B1LTB4R2RXRARXRBRXRG
SCHEMBL8400340 0.89 AKR1B1 (0.46) HTTAKR1B1
SCHEMBL8398941 0.89 AKR1B1 (0.39) AKR1B1LTB4R2
SCHEMBL8395521 0.89 AKR1B1 (0.40) AKR1B1RXRARXRBRXRG
SCHEMBL8396280 0.88 AKR1B1 (0.40) AKR1B1LTB4R2
SCHEMBL8395488 0.88 MTNR1A (0.39) ALDH1A1HTTPAX8AKR1B1LTB4R2
SCHEMBL8400711 0.88 AKR1B1 (0.38) AKR1B1LTB4R2KMT2AMEN1
SCHEMBL8399605 0.87 LTB4R2 (0.39) ALDH1A1HTTPAX8AKR1B1LTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed