SCHEMBL8518906

SCHEMBL8518906

O=C(O)CCC(=O)N(Cc1nc2c(F)c(F)ccc2s1)c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.40
HDAC6 Q9UBN7 3/20 0.39
NOS2 P35228 6/20 0.37
NOS3 P29474 5/20 0.37
LTB4R2 Q9NPC1 1/20 0.36
NOS1 P29475 4/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 1/20 0.36
KCNH2 Q12809 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399142 0.91 AKR1B1 (0.41) AKR1B1LTB4R2
SCHEMBL8400340 0.90 AKR1B1 (0.46) AKR1B1
SCHEMBL8395521 0.89 AKR1B1 (0.40) AKR1B1HDAC6RXRARXRBRXRG
SCHEMBL8400418 0.89 RAB9A (0.40) AKR1B1LTB4R2RXRARXRBRXRG
SCHEMBL8396237 0.88 SMN1; SMN2 (0.40) AKR1B1HDAC6NOS2NOS3LTB4R2
SCHEMBL8397960 0.88 AKR1B1 (0.41) AKR1B1HDAC6LTB4R2
SCHEMBL8398941 0.88 AKR1B1 (0.39) AKR1B1LTB4R2
SCHEMBL8396084 0.87 AKR1A1 (0.46) AKR1B1
SCHEMBL8396327 0.87 AKR1B1 (0.37) AKR1B1HDAC6LTB4R2
SCHEMBL8400428 0.87 AKR1B1 (0.41) AKR1B1HDAC6LTB4R2RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed