SCHEMBL8401430

SCHEMBL8401430

CC(=O)On1c(-c2ccc(F)cc2)ncc(NC(=O)OCc2ccccc2)c1=O

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ELANE P08246 18/20 0.59
MGLL Q99685 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27451145 0.93 ELANE (0.55) ELANEMGLLNPC1RAB9A
SCHEMBL27467025 0.92 ELANE (0.51) ELANENPC1RAB9A
SCHEMBL8401403 0.90 ELANE (0.58) ELANENPC1RAB9A
SCHEMBL8401199 0.90 ELANE (0.59) ELANEMGLLNPC1RAB9A
SCHEMBL8401406 0.89 ELANE (0.50) ELANENPC1RAB9A
SCHEMBL8401266 0.87 ELANE (0.60) ELANENPC1RAB9A
SCHEMBL8405263 0.86 ELANE (0.58) ELANENPC1RAB9A
SCHEMBL27466074 0.85 ELANE (0.46) ELANENPC1RAB9A
SCHEMBL27467469 0.85 NPC1 (0.52) ELANEMGLLNPC1RAB9A
SCHEMBL27448339 0.84 NPC1 (0.53) ELANEMGLLNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188401-C Heterocyclic amide compound and its pharmaceutical use MITSUBISHI PHARMACEUTICAL CO L (JP) 2005-02-09 CN disclosed
CN-1131210-C Heterocyclic amide compound and medical use thereof MITSUBISHI SEIYAKU CO LTD (JP) 2003-12-17 CN disclosed
CN-1088706-C Novel heterocyclic amide compound and medical use thereof MAMORUFUKU KK (JP) 2002-08-07 CN disclosed
CN-1304931-A Heterocyclic amide compound and medical use thereof EFUKU CO LTD (JP) 2001-07-25 CN disclosed
CN-1242014-A Novel heterocyclic amide compounds and medicinal uses thereof YOSHITOMI PHARMACEUTICAL (JP) 2000-01-19 CN disclosed
US-5948785-A USEFUL AS CHYMASE INHIBITORS AND CAN BE EFFECTIVE FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II. THE GREEN CROSS CORPORATION (JP) 1999-09-07 US disclosed
US-5891852-A Serine protease inhibitors-cycloheptane derivatives CORTECH, INC. (US) 1999-04-06 US disclosed
US-5869455-A SUBSTITUTED OXADIAZOLE, THIADIAZOLE AND TRIAZOLE PEPTOIDS WHICH ARE USEFUL AS INHIBITORS OF HUMAN NEUTROPHIL ELASTASE CORTECH, INC. (US) 1999-02-09 US disclosed
US-5861380-A OXADIAZOLE, THIADIAZOLE AND TRIAZOLE PEPTOIDS AS INHIBITORS OF HUMAN NEUTROPHIL ELASTASE; ADULT RESPIRATORY DISTRESS SYNDROME; ANTIARTHRITIC,-INFLAMMATORY,-ISCHEMIC,-TUMOR AND -CARCINOGENIC AGENTS AND OTHER HNE-MEDIATED CONDITIONS CORTECH, INC. (US) 1999-01-19 US disclosed
US-5807829-A RESPIRATORY SYSTEM DISORDERS; SESPIC SHOCK; ORGAN FAILURE CORTECH, INC. (US) 1998-09-15 US disclosed
US-5801148-A Serine protease inhibitors-proline analogs CORTECH, INC. (US) 1998-09-01 US disclosed
CN-1188472-A Heterocyclic amide compound and medical use thereof GREEN CROSS CORP (JP) 1998-07-22 CN disclosed