SCHEMBL8404152

SCHEMBL8404152

CC(=O)SCC=CCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
CASP3 P42574 1/20 0.43
NPC1 O15118 1/20 0.40
GSK3B P49841 1/20 0.40
DRD3 P35462 1/20 0.40
HPGD P15428 2/20 0.39
PLIN1 O60240 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
PLIN5 Q00G26 1/20 0.39
ABHD5 Q8WTS1 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4468251 0.80 CASP3 (0.60) ALDH1A1CA12CA9CASP3DRD3
SCHEMBL8950475 0.80 CASP3 (0.60) ALDH1A1CA12CA9CASP3DRD3
SCHEMBL4476083 0.80 CASP3 (0.60) ALDH1A1CA12CA9CASP3DRD3
SCHEMBL19595059 0.78 CASP3 (0.47) ALDH1A1CA12CA9CASP3NPC1
SCHEMBL16654973 0.78 ALDH1A1 (0.50) ALDH1A1CA12CA9CASP3HPGD
SCHEMBL16654972 0.78 ALDH1A1 (0.50) ALDH1A1CA12CA9CASP3HPGD
SCHEMBL23318802 0.76 NPSR1 (0.48) ALDH1A1CA12CA9CASP3
SCHEMBL28565124 0.76 NPSR1 (0.48) ALDH1A1CA12CA9CASP3
SCHEMBL10176436 0.75 ALDH1A1 (0.42) ALDH1A1CA12CA9CASP3
SCHEMBL9761279 0.75 CASP3 (0.51) ALDH1A1CA12CA9CASP3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0457250-B1 Novel bifunctional linking compounds, conjugates and methods for their production BRISTOL MYERS SQUIBB CO (US) 1999-07-14 EP claimed
EP-0457250-A2 Novel bifunctional linking compounds, conjugates and methods for their production BRISTOL-MYERS SQUIBB COMPANY (US) 1991-11-21 EP claimed
EP-0457250-B1 Novel bifunctional linking compounds, conjugates and methods for their production BRISTOL MYERS SQUIBB CO (US) 1999-07-14 EP disclosed
US-5349066-A Antibodies BRISTOL-MYERS SQUIBB COMPANY (US) 1994-09-20 US disclosed
US-5137877-A N-substituted hydrazine bifuctional derivative; cytotoxic reagent BRISTOL-MYERS SQUIBB (US) 1992-08-11 US disclosed
EP-0457250-A2 Novel bifunctional linking compounds, conjugates and methods for their production BRISTOL-MYERS SQUIBB COMPANY (US) 1991-11-21 EP disclosed