SCHEMBL8405129

SCHEMBL8405129

Cc1cnc(-c2cccnc2)o1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.62
NPC1 O15118 6/20 0.62
RAB9A P51151 6/20 0.62
KDM4E B2RXH2 4/20 0.62
HPGD P15428 4/20 0.62
HSD17B10 Q99714 4/20 0.62
SMN1; SMN2 Q16637 3/20 0.55
CYP2A6 P11509 7/20 0.50
CYP3A4 P08684 4/20 0.50
CYP1A2 P05177 3/20 0.50
CYP2C19 P33261 2/20 0.49
ELANE P08246 1/20 0.49
TP53 P04637 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNA5 P30532 1/20 0.47
CHRNA4 P43681 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL734554 0.80 TSHR (0.59) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL15006930 0.79 NPC1 (0.61) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL13188470 0.78 ALDH1A1 (0.62) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL8405503 0.77 ALDH1A1 (0.62) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL13385756 0.77 TSHR (0.60) ALDH1A1NPC1RAB9AKDM4EHPGD
Bromide SCHEMBL15011830 0.77 NPC1 (0.59) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL4881571 0.76 RAB9A (1.00) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL21408719 0.76 KDM4E (0.41) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL3789884 0.75 KDM4E (0.59) ALDH1A1NPC1RAB9AKDM4EHPGD
SCHEMBL12266934 0.74 RAB9A (0.56) ALDH1A1NPC1RAB9AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7332476-B2 Pyridyl substituted ketolide antibiotics NOVARTIS AG (CH) 2008-02-19 US disclosed
US-7332476-B2 Pyridyl substituted ketolide antibiotics NOVARTIS AG (CH) 2008-02-19 US disclosed
US-RE36374-E 1,2,3-triazole and tetrazole substituted piperidine or tetrahydropyridine compounds useful as acetylcholine agonists H. LUNDBECK, A/S (DK) 1999-11-02 US disclosed
EP-0296721-B1 HETEROCYCLIC COMPOUNDS H. LUNDBECK A/S (DK) 1993-06-23 EP disclosed
US-5053416-A Alzheimer's disease; central cholinomimetic activity ROUSSEL UCLAF (FR) 1991-10-01 US disclosed
EP-0376848-A1 Thiazolyl or oxazolyl substituted 1,2,5,6-tetrahydropyridine derivatives, process and intermediates for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1990-07-04 EP disclosed
US-4925858-A NERVOUS SYSTEM DISORDERS, ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1990-05-15 US disclosed
US-4866077-A TREATMENT OF NERVOUS SYSTEM DISORDERS SUCH AS ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1989-09-12 US disclosed
EP-0296721-A2 Heterocyclic compounds H. LUNDBECK A/S (DK) 1988-12-28 EP disclosed