SCHEMBL8405572

SCHEMBL8405572

COc1cc2c(cc1Br)C(C)NCC2

nearest known ligand 0.77

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOA P21397 8/20 0.77
TSHR P16473 2/20 0.77
HTR2C P28335 7/20 0.67
HTR2B P41595 7/20 0.67
HTR2A P28223 6/20 0.67
HSD17B10 Q99714 2/20 0.64
CYP2D6 P10635 1/20 0.64
ALDH1A1 P00352 1/20 0.64
DRD2 P14416 2/20 0.53
KDM4E B2RXH2 1/20 0.53
CYP2C9 P11712 1/20 0.53
DRD3 P35462 1/20 0.53
HIF1A Q16665 1/20 0.53
DRD4 P21917 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7847453 0.94 MAOA (0.77) MAOATSHRHTR2CHTR2BHTR2A
Salsolidine SCHEMBL1819825 0.87 MAOA (1.00) MAOATSHRHSD17B10CYP2D6ALDH1A1
Salsolidine SCHEMBL4250569 0.87 MAOA (1.00) MAOATSHRHSD17B10CYP2D6ALDH1A1
Salsolidine SCHEMBL34461883 0.87 MAOA (1.00) MAOATSHRHSD17B10CYP2D6ALDH1A1
Salsolidine SCHEMBL177753 0.87 MAOA (1.00) MAOATSHRHSD17B10CYP2D6ALDH1A1
Salsolidine SCHEMBL7838872 0.85 MAOA (0.97) MAOATSHRHSD17B10CYP2D6ALDH1A1
Salsolidine SCHEMBL5242077 0.85 MAOA (1.00) MAOATSHRHSD17B10CYP2D6ALDH1A1
SCHEMBL1009124 0.83 MAOA (0.62) MAOATSHRHTR2CHTR2BHTR2A
SCHEMBL1094326 0.80 HTR2C (1.00) HTR2CHTR2BHTR2A
SCHEMBL1094962 0.80 HTR2C (1.00) HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981521-A USEFUL FOR TREATING VARIOUS HORMONE DEPENDENT DISEASES, INCLUDING PROSTATE CANCER, ENDOMETRIOSIS, UTERINE FIBROIDS, PRECOCIOUS PUBERTY, BENIGN PROSTATE HYPERTROPY AND IN VITRO FERTILIZATION ABBOTT LABORATORIES (US) 1999-11-09 US disclosed