SCHEMBL8405741

SCHEMBL8405741

Cc1ccc(CC(=O)n2cncc(NC(=O)OCc3ccccc3)c2=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
ELANE P08246 5/20 0.42
OPRK1 P41145 2/20 0.41
MAPT P10636 1/20 0.41
CASP3 P42574 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
SCD O00767 1/20 0.41
CTRC Q99895 1/20 0.41
FAAH O00519 1/20 0.40
MGLL Q99685 1/20 0.40
P2RX3 P56373 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297137 0.94 NPC1 (0.48) NPC1RAB9APOLBSMN1; SMN2ELANE
SCHEMBL8401497 0.91 NPC1 (0.47) TRPV1NPC1RAB9APOLBSMN1; SMN2
SCHEMBL8401151 0.90 ELANE (0.46) NPC1RAB9APOLBSMN1; SMN2ELANE
SCHEMBL7292947 0.90 ELANE (0.45) NPC1RAB9APOLBSMN1; SMN2ELANE
SCHEMBL8403664 0.90 SCD (0.48) TRPV1NPC1RAB9APOLBSMN1; SMN2
SCHEMBL8401233 0.90 POLB (0.53) TRPV1NPC1RAB9APOLBELANE
SCHEMBL8405275 0.87 NPC1 (0.53) TRPV1NPC1RAB9APOLBSMN1; SMN2
SCHEMBL7294413 0.87 NAMPT (0.47) TRPV1NPC1RAB9APOLBELANE
SCHEMBL8405850 0.86 ELANE (0.47) NPC1RAB9APOLBELANE
SCHEMBL7293123 0.82 HDAC3 (0.44) NPC1RAB9APOLBELANEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948785-A USEFUL AS CHYMASE INHIBITORS AND CAN BE EFFECTIVE FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II. THE GREEN CROSS CORPORATION (JP) 1999-09-07 US disclosed