SCHEMBL8406937

SCHEMBL8406937

COC(=O)c1cccnc1N(C)C1CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CNR2 P34972 1/20 0.41
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
KDM4E B2RXH2 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
PKM P14618 1/20 0.38
HTR2C P28335 1/20 0.38
OPRK1 P41145 4/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
KCNH2 Q12809 1/20 0.37
GCK P35557 1/20 0.37
PCSK9 Q8NBP7 2/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12516141 0.80 KMT2A (0.43) ADRA1DADRA1AADRA1BOPRK1SLC6A2
SCHEMBL2223213 0.80 KMT2A (0.43) ADRA1DADRA1AADRA1BOPRK1SLC6A2
SCHEMBL2222662 0.80 KMT2A (0.43) ADRA1DADRA1AADRA1BOPRK1SLC6A2
Hydrochloric Acid SCHEMBL2222676 0.79 KMT2A (0.42) ADRA1DADRA1AADRA1BOPRK1SLC6A2
SCHEMBL8406740 0.78 DRD2 (0.62) ALDH1A1TDP1KDM4EL3MBTL1PKM
SCHEMBL3716902 0.74 PARP1 (0.44) ALDH1A1TDP1KDM4EKCNH2
SCHEMBL3714492 0.73 JAK3 (0.43) ALDH1A1KDM4EKCNH2
SCHEMBL8408485 0.73 DRD2 (0.46) ALDH1A1TDP1SLC6A2SLC6A4
SCHEMBL20545619 0.73 TDP1 (0.49) MAP2K1ALDH1A1TDP1CNR2KDM4E
SCHEMBL21119052 0.72 ALDH1A1 (0.51) ALDH1A1TDP1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed