SCHEMBL8407940

SCHEMBL8407940

COC(=O)Nc1c(F)cccc1OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.54
RAB9A P51151 4/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
BRD4 O60885 2/20 0.51
MRGPRX4 Q96LA9 1/20 0.51
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
CASP3 P42574 3/20 0.50
SENP7 Q9BQF6 3/20 0.50
KDM4E B2RXH2 1/20 0.50
KDM1A O60341 2/20 0.47
SGMS2 Q8NHU3 1/20 0.47
PPIA P62937 2/20 0.46
MAPT P10636 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TAAR1 Q96RJ0 1/20 0.45
LMNA P02545 1/20 0.45
HTR1A P08908 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431920 0.89 NPC1 (0.54) NPC1RAB9ASMN1; SMN2BRD4MRGPRX4
SCHEMBL2894833 0.87 NPC1 (0.50) NPC1RAB9ASMN1; SMN2BRD4MRGPRX4
SCHEMBL2892753 0.82 NPC1 (0.52) NPC1RAB9ASMN1; SMN2BRD4MRGPRX4
Hydrochloric Acid SCHEMBL28557881 0.78 NPC1 (0.48) NPC1RAB9ASMN1; SMN2BRD4MRGPRX4
SCHEMBL8405081 0.77 NPC1 (0.53) NPC1RAB9ASMN1; SMN2BRD4MRGPRX4
SCHEMBL4825037 0.77 NLRP3 (0.58) RAB9ASMN1; SMN2MEN1KMT2AL3MBTL1
SCHEMBL21862932 0.75 NPC1 (0.45) NPC1RAB9ABRD4MRGPRX4MEN1
SCHEMBL27724257 0.74 NPC1 (0.53) NPC1RAB9ABRD4MRGPRX4MEN1
SCHEMBL2897224 0.74 MRGPRX4 (0.62) NPC1MRGPRX4MEN1KMT2AKDM1A
SCHEMBL27849246 0.74 NPC1 (0.52) NPC1RAB9ASMN1; SMN2BRD4MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624567-B1 Derivatives of 3-fluorophenol, process for their preparation and their use CLARIANT GMBH (DE) 1999-12-08 EP disclosed
EP-0628536-B1 Process for the preparation of aromatic amines CLARIANT GMBH (DE) 1999-07-14 EP disclosed
US-5410082-A Process for preparing amines CLARIANT GMBH (DE) 1995-04-25 US disclosed
EP-0628536-A2 Process for the preparation of amines HOECHST AKTIENGESELLSCHAFT (DE) 1994-12-14 EP disclosed
EP-0624567-A2 Derivatives of 3-fluorophenol, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1994-11-17 EP disclosed