SCHEMBL8408602

SCHEMBL8408602

N#Cc1ccc(C(CCc2ccc(F)cc2)c2nnn[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.52
CACNA1F O60840 2/20 0.42
HTR1A P08908 2/20 0.42
ADORA3 P0DMS8 2/20 0.42
DRD2 P14416 2/20 0.42
DRD1 P21728 2/20 0.42
DRD4 P21917 2/20 0.42
DRD5 P21918 2/20 0.42
HRH2 P25021 2/20 0.42
ADRA1D P25100 2/20 0.42
HTR2A P28223 2/20 0.42
HTR7 P34969 2/20 0.42
ADRA1A P35348 2/20 0.42
HRH1 P35367 2/20 0.42
ADRA1B P35368 2/20 0.42
OPRM1 P35372 2/20 0.42
DRD3 P35462 2/20 0.42
HTR6 P50406 2/20 0.42
CACNA1D Q01668 2/20 0.42
SLC6A3 Q01959 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9196337 0.82 CYP19A1 (0.56) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL8408610 0.80 CYP19A1 (0.54) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL8410909 0.75 CYP19A1 (0.54) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL8411281 0.73 CYP19A1 (0.63) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL8109000 0.72 CYP19A1 (0.54) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL9194497 0.72 CYP19A1 (0.54) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL8104816 0.72 CYP19A1 (0.54) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL5597463 0.71 CYP19A1 (0.51) CYP19A1OPRD1
SCHEMBL9089515 0.69 CYP19A1 (0.64) CYP19A1CACNA1FHTR1AADORA3DRD2
SCHEMBL8408857 0.68 CYP19A1 (0.63) CYP19A1CACNA1FHTR1AADORA3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674626-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS ORION-YHTYMÄ OY (FI) 1995-10-04 EP claimed
US-5962495-A ESTROGEN SENSITIVE DISEASES; BREAST CANCER; PROSTATE TUMORS RISTO ARVO SAKARI LAMMINTAUSTA (FI) 1999-10-05 US disclosed
US-5703109-A CYANOPHENYL-1,2,4-TRIAZOLE DERIVATIVE Oy, Orion-yhtyma (FI) 1997-12-30 US disclosed
EP-0674626-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS ORION-YHTYMÄ OY (FI) 1995-10-04 EP disclosed