SCHEMBL8409288

SCHEMBL8409288

COC(=O)CCCCS(=O)(=O)c1ccc(-c2ccc(C#N)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.49
HDAC2 Q92769 3/20 0.49
MMP3 P08254 6/20 0.45
MMP2 P08253 6/20 0.43
MMP13 P45452 6/20 0.43
MMP1 P03956 5/20 0.43
MMP9 P14780 5/20 0.43
MMP7 P09237 4/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
EGLN1 Q9GZT9 1/20 0.41
KDM1A O60341 1/20 0.40
ACLY P53396 1/20 0.40
ADAMTS4 O75173 1/20 0.40
CYP19A1 P11511 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713200 0.96 HDAC1 (0.43) HDAC1HDAC2MMP1CA12CA1
SCHEMBL8407563 0.81 ALDH1A1 (0.56) HDAC1HDAC2MMP3MMP2MMP13
SCHEMBL9703247 0.80 HDAC1 (0.61) HDAC1HDAC2MMP3MMP2MMP13
SCHEMBL8886240 0.79 CYP19A1 (0.47) MMP3MMP2MMP13MMP1MMP9
SCHEMBL4711012 0.79 KMT2A (0.47) MMP1CYP19A1ALDH1A1
SCHEMBL8410478 0.79 MMP3 (0.71) HDAC1HDAC2MMP3MMP2MMP13
SCHEMBL8409326 0.79 CYP11B1 (0.43) HDAC1HDAC2MMP3MMP2MMP13
SCHEMBL8779427 0.78 ALDH1A1 (0.59) HDAC1HDAC2CA12CA1CA2
SCHEMBL17045867 0.78 HDAC1 (0.49) HDAC1HDAC2MMP13MMP1CA2
SCHEMBL19183052 0.78 KDM1A (0.48) MMP3MMP2MMP13MMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed