SCHEMBL8409443

SCHEMBL8409443

COC(=O)CN1CCN(C(=O)c2ccc(-c3ccc(C#N)cc3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 1/20 0.54
KCNA5 P22460 1/20 0.52
USP2 O75604 2/20 0.49
CYP2C9 P11712 2/20 0.49
TSHR P16473 2/20 0.49
CYP1A2 P05177 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49
PTGER4 P35408 1/20 0.48
PTGER2 P43116 1/20 0.48
PTGDR Q13258 1/20 0.48
CYP3A4 P08684 3/20 0.48
CYP2D6 P10635 1/20 0.48
MKNK1 Q9BUB5 3/20 0.47
MKNK2 Q9HBH9 3/20 0.47
NOS1 P29475 1/20 0.47
NOS2 P35228 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408009 0.88 KCNA5 (0.56) SLC6A7KCNA5USP2CYP2C9TSHR
SCHEMBL15557487 0.84 KCNA5 (0.53) SLC6A7KCNA5USP2CYP2C9TSHR
SCHEMBL8410628 0.81 PTGER4 (0.54) SLC6A7USP2CYP2C9TSHRCYP1A2
SCHEMBL8407569 0.81 CCNK (0.51) SLC6A7USP2CYP2C9TSHRCYP1A2
Hydrochloric Acid SCHEMBL8714344 0.81 KDM1A (0.54) ALDH1A1DRD2MEN1KMT2ADRD3
SCHEMBL15557338 0.79 KCNA5 (0.52) SLC6A7KCNA5USP2CYP2C9TSHR
SCHEMBL16627284 0.79 KCNA5 (0.68) KCNA5USP2CYP2C9TSHRCYP1A2
SCHEMBL9171577 0.78 POLB (0.59) KCNA5SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL19634410 0.77 DRD2 (0.50) HRH3ALDH1A1DRD2MEN1KMT2A
SCHEMBL8560134 0.77 KDM1A (0.49) NOS1NOS2ALDH1A1CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed