SCHEMBL8560134

SCHEMBL8560134

COC(=O)CC1CCN(C(=O)c2ccc(-c3ccc(C#N)cc3)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 11/20 0.49
ALDH1A1 P00352 1/20 0.48
EGLN1 Q9GZT9 1/20 0.47
CCNK O75909 1/20 0.47
CDK12 Q9NYV4 1/20 0.47
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
GRM3 Q14832 3/20 0.46
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720191 0.94 GRM3 (0.54) KDM1AALDH1A1GRM3
SCHEMBL8407569 0.93 CCNK (0.51) KDM1AALDH1A1CCNKCDK12NOS1
SCHEMBL8407511 0.85 MLNR (0.46) KDM1AALDH1A1
SCHEMBL8410939 0.83 GRM3 (0.50) KDM1AALDH1A1GRM3
SCHEMBL8719948 0.82 KDM1A (0.49) KDM1AALDH1A1CCNKCDK12NOS1
Hydrochloric Acid SCHEMBL8407950 0.82 ITGB3 (0.46)
SCHEMBL8949062 0.82 CCNK (0.47) EGLN1CCNKCDK12NOS1NOS2
SCHEMBL8718956 0.80 MLNR (0.48) KDM1AALDH1A1
SCHEMBL8409445 0.80 CHRM4 (0.52) KDM1AALDH1A1CCNKCDK12
SCHEMBL8407175 0.79 GAA (0.47) KDM1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed