SCHEMBL8409651

SCHEMBL8409651

c1ccc(Oc2ccc(-c3nc4cc(C5=NCCN5)ccc4[nH]3)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.64
MAOA P21397 1/20 0.53
MAOB P27338 1/20 0.53
CHEK2 O96017 5/20 0.52
PRMT1 Q99873 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13204584 0.85 NISCH (0.54) NISCHPRMT1
SCHEMBL9241934 0.84 CHEK2 (0.66) CHEK2
SCHEMBL8141749 0.79 NISCH (1.00) NISCHMAOAMAOB
SCHEMBL548343 0.79 NISCH (0.50) NISCHMAOBPRMT1
SCHEMBL549218 0.79 TOP2A (0.56) NISCHPRMT1
SCHEMBL8677423 0.79 NISCH (0.50) NISCHMAOBPRMT1
SCHEMBL548359 0.79 NISCH (0.52) NISCHPRMT1
SCHEMBL8477890 0.79 NPC1 (0.58) NISCHPRMT1
SCHEMBL14599548 0.78 PRMT1 (0.49) NISCHPRMT1
SCHEMBL14599545 0.77 NISCH (0.48) NISCHPRMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942532-A INHIBITORS OF HISTIDINE PROTEIN KINASE; BACTERIA RESISTANT TO OTHER ANTIBIOTICS ORTHO PHARMACEUTICAL CORPORATION (US) 1999-08-24 US disclosed
WO-1999011627-A1 2-SUBSTITUTED PHENYL-BENZIMIDAZOLE ANTIBACTERIAL AGENTS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 1999-03-11 WO disclosed