SCHEMBL8409833

SCHEMBL8409833

CCNc1cccnc1N(CC)CC1CCNCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 3/20 0.37
IDO1 P14902 1/20 0.36
CXCR4 P61073 4/20 0.35
CYP2D6 P10635 2/20 0.35
GRM5 P41594 1/20 0.33
AXL P30530 1/20 0.33
FLT3 P36888 1/20 0.33
TYRO3 Q06418 1/20 0.33
MERTK Q12866 1/20 0.33
GAS6 Q14393 1/20 0.33
TP53 P04637 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
FFAR2 O15552 2/20 0.32
BRD4 O60885 1/20 0.31
ATAD2 Q6PL18 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8409811 0.86 KHK (0.36) KHKCXCR4CYP2D6AXLFLT3
SCHEMBL8407524 0.86 KHK (0.36) KHKIDO1CXCR4CYP2D6AXL
SCHEMBL8791217 0.81 KHK (0.39) KHKCXCR4CYP2D6TP53FFAR2
SCHEMBL8406794 0.80 SLC6A2 (0.40) IDO1GRM5TP53ADRA1DADRA1A
SCHEMBL10606573 0.80 IDO1 (0.47) IDO1GRM5
SCHEMBL8409924 0.79 ACHE (0.49) CYP2D6TP53
SCHEMBL9093069 0.77 DRD2 (0.38) TYRO3
SCHEMBL8406705 0.76 TP53 (0.37) IDO1GRM5TP53PTK2
SCHEMBL9640162 0.72 IDO1 (0.44) IDO1GRM5
SCHEMBL8408425 0.71 SLC6A2 (0.39) KHKAXLFLT3TYRO3MERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed