SCHEMBL8411503

SCHEMBL8411503

CC(CSCCC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
APEX1 P27695 1/20 0.35
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
PPARG P37231 3/20 0.32
PPARA Q07869 3/20 0.32
NOS1 P29475 2/20 0.31
NOS2 P35228 2/20 0.31
NOS3 P29474 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15082197 1.00 HDAC3 (0.38) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL15490645 0.83 CYP1A2 (0.42) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL8414944 0.81 HDAC3 (0.39) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL22110077 0.81 TSHR (0.43) APEX1CYP1A2MEN1KMT2ANOS1
SCHEMBL5014070 0.80 HDAC1 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL17632961 0.79 DGKA (0.36) APEX1CYP1A2KMT2ANOS1NOS2
SCHEMBL12171658 0.77 CYP1A2 (0.54) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL18134688 0.77 CYP1A2 (0.54) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL5014073 0.77 LMNA (0.56) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL17227860 0.77 CYP1A2 (0.54) HDAC3HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0932598-A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1999-08-04 EP disclosed
WO-1998016502-A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1998-04-23 WO disclosed