SCHEMBL8411729

SCHEMBL8411729

NC#CC(=O)OC1CCCCCC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.42
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
STS P08842 4/20 0.38
CYP2C19 P33261 1/20 0.38
CA12 O43570 2/20 0.38
CA9 Q16790 2/20 0.38
NAAA Q02083 2/20 0.37
HTT P42858 1/20 0.36
CYP19A1 P11511 3/20 0.36
MMP1 P03956 1/20 0.33
MMP9 P14780 1/20 0.33
MMP12 P39900 1/20 0.33
FABP7 O15540 1/20 0.33
FABP5 Q01469 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2531983 0.87 EPHX1 (0.48) EPHX1CA1CA2STSCYP2C19
SCHEMBL2528803 0.84 EPHX1 (0.45) EPHX1CA1CA2STSCYP2C19
SCHEMBL25333252 0.79 EPHX1 (0.42) EPHX1CA1CA2STSCYP2C19
SCHEMBL733037 0.76 EPHX1 (0.47) EPHX1CA1CA2STSCYP2C19
SCHEMBL31339503 0.74 EPHX1 (0.45) EPHX1CA1CA2STSCYP2C19
SCHEMBL27981763 0.74 EPHX1 (0.45) EPHX1CA1CA2STSCYP2C19
SCHEMBL31339498 0.74 EPHX1 (0.45) EPHX1CA1CA2STSCYP2C19
SCHEMBL6207813 0.74 EPHX1 (0.45) EPHX1CA1CA2STSCYP2C19
SCHEMBL11473389 0.74 EPHX1 (0.45) EPHX1CA1CA2STSCYP2C19
SCHEMBL27567894 0.72 NAAA (0.46) EPHX1CA1CA2STSCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
EP-0591040-B1 Quaternary basic amides as tachykinines antagonists SANOFI SA (FR) 1999-02-03 EP disclosed
EP-0591040-A1 Quaternary basic amides as tachykinines antagonists SANOFI (FR) 1994-04-06 EP disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed