Nimustine

Nimustine

SCHEMBL8414

Cc1ncc(CNC(=O)N(CCCl)N=O)c(N)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BLM P54132 2/20 1.00
PMP22 Q01453 2/20 1.00
LMNA P02545 2/20 1.00
NFKB1 P19838 1/20 1.00
ALDH1A1 P00352 2/20 0.45
TSHR P16473 2/20 0.45
MEN1 O00255 1/20 0.45
ABCB11 O95342 1/20 0.45
GSR P00390 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
ADRA2A P08913 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35
TKT P29401 4/20 0.35
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nimustine SCHEMBL23301409 1.00 BLM (1.00) BLMPMP22LMNANFKB1ALDH1A1
Nimustine SCHEMBL98303 0.99 BLM (0.98) BLMPMP22LMNANFKB1ALDH1A1
Nimustine SCHEMBL1649545 0.99 BLM (0.98) BLMPMP22LMNANFKB1ALDH1A1
Nimustine SCHEMBL124427 0.99 BLM (0.98) BLMPMP22LMNANFKB1ALDH1A1
Nimustine SCHEMBL1649348 0.98 BLM (0.96) BLMPMP22LMNANFKB1ALDH1A1
Nimustine SCHEMBL1580335 0.96 BLM (0.92) BLMPMP22LMNANFKB1ALDH1A1
Nimustine SCHEMBL5886061 0.89 BLM (0.80) BLMPMP22LMNANFKB1ALDH1A1
SCHEMBL25299723 0.88 LMNA (0.79) BLMPMP22LMNANFKB1TKT
SCHEMBL17524414 0.88 BLM (0.79) BLMPMP22LMNANFKB1ALDH1A1
SCHEMBL6541875 0.83 LMNA (0.71) BLMPMP22LMNANFKB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 42533 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
US-20260137700-A1 PHARMACEUTICAL COMBINATION OF PRMT5 INHIBITOR AND DNA DAMAGE-INDUCING SUBSTANCE SK BIOPHARMACEUTICALS CO LTD (KR) 2026-05-21 US claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026101232-A1 POLYMER COMPOUND FOR CELL SURFACE MODIFICATION FOR IMPROVING DRUG DELIVERY EFFICIENCY 동국대학교 산학협력단 2026-05-15 WO claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
WO-2025136820-A9 POLY-ANTIGEN CYTOKINE-RECEPTOR COMPLEXES (PACCS), COMPOSITIONS, AND METHODS OF USE REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2026-05-15 WO claimed
CN-122011207-A CAR-T cell over-expressing H2A.Z as well as preparation method and application thereof 中国科学院微生物研究所 2026-05-12 CN claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-4103170-B1 A PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF A CANCER ABILITY PHARMACEUTICALS S A (ES) 2026-04-08 EP claimed
US-20260091119-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF GLIOMA CELLIS AG (CH) 2026-04-02 US claimed
EP-0977725-A1 NEW FATTY ACID DERIVATIVES NORSK HYDRO ASA (NO) 2000-02-09 EP claimed
WO-1999058126-A1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1999-11-18 WO claimed
WO-1999042578-A2 MODULATION OF CELL PROLIFERATION, METHODS AND REAGENTS COLD SPRING HARBOR LABORATORY (US) 1999-08-26 WO claimed
WO-1998032718-A1 NEW FATTY ACID DERIVATIVES NORSK HYDRO ASA (NO) 1998-07-30 WO claimed
US-5756475-A POLYISOPRENE MODIFIED WITH AMINE WITH ANTICANCER AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-26 US claimed
US-5691307-A ANTITUMOR AGENTS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1997-11-25 US claimed
EP-0758249-A1 PROGRAMMABLE GENOTOXIC AGENTS AND USES THEREFOR MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1997-02-19 EP claimed
WO-1995030442-A1 PROGRAMMABLE GENOTOXIC AGENTS AND USES THEREFOR MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1995-11-16 WO claimed
EP-0174342-B1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1989-12-20 EP claimed
US-4003901-A ANTILEUKEMIA SANKYO COMPANY LIMITED (JA) 1977-01-18 US claimed