SCHEMBL8417822

SCHEMBL8417822

CC(C)(C)OC(=O)NCc1ccc(O)c(C(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.53
KLKB1 P03952 1/20 0.51
CTSB P07858 1/20 0.51
MMP9 P14780 1/20 0.51
DNMT1 P26358 1/20 0.51
DNMT3B Q9UBC3 1/20 0.51
DNMT3L Q9UJW3 1/20 0.51
DNMT3A Q9Y6K1 1/20 0.51
LCK P06239 2/20 0.48
HNF4A P41235 1/20 0.47
KAT8 Q9H7Z6 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
NAMPT P43490 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
NR1H4 Q96RI1 2/20 0.43
GAA P10253 1/20 0.43
KDM4A O75164 1/20 0.43
HPN P05981 1/20 0.43
KDM4C Q9H3R0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30910306 0.89 NR1H4 (0.48) HDAC1L3MBTL1NAMPTCA1CA2
SCHEMBL1205128 0.89 NR1H4 (0.48) HDAC1L3MBTL1NAMPTCA1CA2
SCHEMBL8417963 0.88 HPN (0.49) HDAC1L3MBTL1NAMPTCA1CA2
SCHEMBL14979282 0.87 NR1H4 (0.50) HDAC1L3MBTL1NAMPTCA1CA2
SCHEMBL30901987 0.87 NR1H4 (0.50) HDAC1L3MBTL1NAMPTCA1CA2
SCHEMBL5749285 0.85 ERCC1 (0.56) HDAC1LCKL3MBTL1NAMPTCA1
SCHEMBL1671124 0.85 TSHR (0.55) HDAC1L3MBTL1NAMPTNR1H4GAA
SCHEMBL6625230 0.85 NR1H4 (0.50) HDAC1L3MBTL1NAMPTNR1H4GAA
SCHEMBL474132 0.85 ALDH1A1 (0.53) HDAC1L3MBTL1NAMPTCA1CA2
SCHEMBL16415399 0.85 HDAC1 (0.47) HDAC1L3MBTL1NAMPTCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922697-A Compounds, compositions and methods for inhibiting the binding of proteins containing an SH2 domain to cognate phosphorylated proteins WARNER-LAMBERT COMPANY (US) 1999-07-13 US disclosed
WO-1997012903-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR INHIBITING THE BINDING OF PROTEINS CONTAINING AN SH2 DOMAIN TO COGNATE PHOSPHORYLATED PROTEINS WARNER-LAMBERT COMPANY (US) 1997-04-10 WO disclosed