SCHEMBL8420730

SCHEMBL8420730

CS(=O)(=O)c1ccc(-n2nc(-c3ccc(Br)cc3)cc2-c2ccc(Br)cc2)cc1

nearest known ligand 0.88

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.88
MMP2 P08253 1/20 0.58
RARA P10276 3/20 0.57
RARB P10826 3/20 0.57
RARG P13631 3/20 0.57
RXRA P19793 3/20 0.57
ALOX5 P09917 1/20 0.56
CYP2C9 P11712 2/20 0.56
PTGS1 P23219 1/20 0.55
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
USP8 P40818 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420724 0.94 PTGS2 (0.79) PTGS2MMP2RARARARBRARG
SCHEMBL8420040 0.94 PTGS2 (0.79) PTGS2MMP2RARARARBRARG
SCHEMBL8420247 0.88 CYP2C9 (0.71) PTGS2RARARARBRARGRXRA
SCHEMBL8421924 0.86 PTGS2 (0.72) PTGS2RARARARBRARGRXRA
SCHEMBL8121677 0.86 PTGS2 (0.88) PTGS2MMP2CYP2C9PTGS1CA1
SCHEMBL8421061 0.86 PTGS2 (0.88) PTGS2RARARARBRARGRXRA
SCHEMBL8420804 0.86 PTGS2 (0.88) PTGS2RARARARBRARGRXRA
SCHEMBL5215929 0.86 PTGS2 (0.82) PTGS2RARARARBRARGRXRA
SCHEMBL8421888 0.84 PTGS2 (0.71) PTGS2PTGS1CA1CA2
SCHEMBL8421797 0.84 PTGS2 (0.65) PTGS2RARARARBRARGRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed