SCHEMBL8421963

SCHEMBL8421963

CS(=O)(=O)c1ccc(-n2nc(-c3ccc(C#N)cc3)cc2-c2ccc(C#N)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.64
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
RARA P10276 4/20 0.54
RARB P10826 4/20 0.54
RARG P13631 4/20 0.54
RXRA P19793 4/20 0.54
ALOX5 P09917 1/20 0.53
CYP2C9 P11712 2/20 0.53
PTGS1 P23219 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8424138 0.94 PTGS2 (0.74) PTGS2CA1CA2CA9RARA
SCHEMBL8420699 0.94 PTGS2 (0.74) PTGS2CA1CA2CA9RARA
SCHEMBL7459996 0.88 PTGS2 (0.62) PTGS2CA1CA2CA9ALOX5
SCHEMBL8122646 0.88 PTGS2 (0.71) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8420327 0.84 PTGS2 (0.67) PTGS2RARARARBRARGRXRA
SCHEMBL7466476 0.84 PTGS2 (0.74) PTGS2CA1CA2CA9ALOX5
SCHEMBL8420247 0.84 CYP2C9 (0.71) PTGS2CA1CA2CA9RARA
SCHEMBL8421916 0.84 PTGS2 (0.66) PTGS2RARARARBRARGRXRA
SCHEMBL14857165 0.83 PTGS2 (0.80) PTGS2CA1CA2CA9PTGS1
SCHEMBL8421061 0.83 PTGS2 (0.88) PTGS2RARARARBRARGRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed