SCHEMBL8422295

SCHEMBL8422295

Cc1ccc(-c2cc(-c3ccc(Cl)cc3)nn2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.47
MAPT P10636 3/20 0.47
NPY5R Q15761 1/20 0.47
KDM1A O60341 3/20 0.44
MAOA P21397 2/20 0.44
PTGS2 P35354 3/20 0.43
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
PTGES O14684 1/20 0.42
ALOX5 P09917 1/20 0.42
TP53 P04637 1/20 0.41
AURKA O14965 1/20 0.41
MALT1 Q9UDY8 3/20 0.41
PPP1CA P62136 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026973 1.00 CYP2C9 (0.47) CYP2C9MAPTNPY5RKDM1AMAOA
SCHEMBL8420749 0.94 MAPT (0.52) CYP2C9MAPTNPY5RPTGS2SMN1; SMN2
SCHEMBL8421776 0.94 KDM1A (0.47) MAPTKDM1AMAOAPTGS2GAA
SCHEMBL8641119 0.93 AURKA (0.46) CYP2C9MAPTKDM1AMAOAPTGS2
SCHEMBL8421504 0.92 MALT1 (0.40) CYP2C9MAPTNPY5RKDM1AMAOA
SCHEMBL8423750 0.90 KDM1A (0.46) CYP2C9MAPTNPY5RKDM1AMAOA
SCHEMBL8422282 0.90 KDM1A (0.43) CYP2C9MAPTNPY5RKDM1AMAOA
SCHEMBL8424131 0.89 KDM1A (0.41) MAPTNPY5RKDM1AMAOAPTGS2
SCHEMBL8421856 0.89 KDM1A (0.41) MAPTNPY5RKDM1AMAOAPTGS2
SCHEMBL8422285 0.88 MAPT (0.43) MAPTNPY5RKDM1AMAOAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed