SCHEMBL842236

SCHEMBL842236

CC(=O)c1ccc(N)c(Br)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.52
CREBBP Q92793 1/20 0.47
CA2 P00918 2/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
CA5A P35218 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CA5B Q9Y2D0 1/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 5/20 0.42
MAPK1 P28482 2/20 0.42
HTT P42858 1/20 0.42
CYP2A6 P11509 1/20 0.41
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30468765 1.00 PRKCI (0.52) PRKCICREBBPCA2CA12CA1
SCHEMBL7109894 0.83 PRKCI (0.56) PRKCICREBBPCA2NPC1RAB9A
SCHEMBL1376911 0.83 ALDH1A1 (0.52) CA2CA12CA1CA4CA6
SCHEMBL1008508 0.81 CDC25B (0.55) CA2CA12CA1CA4CA6
SCHEMBL30508415 0.81 PRKCI (0.53) PRKCICREBBPNPC1RAB9ASMN1; SMN2
SCHEMBL3090722 0.81 PARP1 (0.50) CA2CA12CA1CA4CA6
SCHEMBL1026788 0.81 PRKCI (0.53) PRKCICREBBPNPC1RAB9ASMN1; SMN2
SCHEMBL265937 0.80 PRKCI (0.62) PRKCICREBBPNPC1RAB9AMAPT
SCHEMBL3022646 0.80 MAPT (0.47) PRKCINPC1RAB9ASMN1; SMN2MAPT
SCHEMBL31495791 0.80 PRKCI (0.62) PRKCICREBBPNPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 95 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4558485-A1 TEAD INHIBITORS AND METHODS OF USE Sporos Biodiscovery, Inc. (US) 2025-05-28 EP disclosed
CN-119497708-A TEAD inhibitors and methods of use 思博睿生物探索公司 2025-02-21 CN disclosed
US-20250026721-A1 COMPOUNDS AND METHODS FOR MODULATING RAS-PI3K VIVIDION THERAPEUTICS, INC. 2025-01-23 US disclosed
WO-2024020350-A1 TEAD INHIBITORS AND METHODS OF USE SPOROS BIODISCOVERY, INC. (US) 2024-01-25 WO disclosed
WO-2024020350-A1 TEAD INHIBITORS AND METHODS OF USE SPOROS BIODISCOVERY, INC. (US) 2024-01-25 WO disclosed
CN-113845548-B Platinum complex of quinazoline hydrazine dithioformate and preparation method and application thereof 深圳大学 2023-06-06 CN disclosed
WO-2022224223-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CORONAVIRAL RELATED DISEASES NOVARTIS AG (CH) 2022-10-27 WO disclosed
CN-109912434-B Synthesis method of phenylethanolamine beta receptor agonist 上海安谱实验科技股份有限公司 2022-07-12 CN disclosed
CN-109912434-A The synthetic method of phenyl ethyl amine beta receptor agonist 上海安谱实验科技股份有限公司 2019-06-21 CN disclosed
EP-3040329-B1 AROMATIC COMPOUND AND USE THEREOF IN THE TREATMENT OF DISORDERS ASSOCIATED WITH BONE METABOLISM KYOTO PHARMA IND (JP) 2018-10-10 EP disclosed
WO-1997035539-A2 ARYLAMINO FUSED PYRIDINES AND PYRIMIDINES DU PONT PHARMACEUTICALS COMPANY (US) 1997-10-02 WO disclosed
US-4814350-A HYPOGLYCEMIC AMERICAN CYANAMID COMPANY (US) 1989-03-21 US disclosed
US-4754047-A ANIMAL GROWTH REGULATORS AMERICAN CYANAMID COMPANY (US) 1988-06-28 US disclosed
EP-0260400-A2 Method of treating diabetes with 5-[1-hydroxy-2-(isopropylamino)-ethyl]anthranilonitrile AMERICAN CYANAMID COMPANY (US) 1988-03-23 EP disclosed
EP-0049728-B1 METHOD FOR ENHANCING THE GROWTH RATE OF MEAT-PRODUCING ANIMALS AND FOR IMPROVING THE LEAN MEAT TO FAT RATIO THEREOF AMERICAN CYANAMID COMPANY (US) 1986-11-12 EP disclosed
US-4522822-A Phenylethane derivatives and acid addition salts thereof for increasing lean meat deposition and/or improving lean meat to fat ratio in warm blooded animals AMERICAN CYANAMID COMPANY (US) 1985-06-11 US disclosed
US-4501751-A Phenylethanolamine derivatives and acid addition salts thereof for enhancing the growth rate of meat-producing animals and improving the efficiency of feed utilization thereby AMERICAN CYANAMID COMPANY (US) 1985-02-26 US disclosed
US-4407819-A ANIMAL GROWTH REGULATORS AMERICAN CYANAMID COMPANY (US) 1983-10-04 US disclosed
US-4404222-A Phenylethanolamine derivatives and acid addition salts thereof for enhancing the growth rate of meat-producing animals and improving the efficiency of feed utilization thereby AMERICAN CYANAMID COMPANY (US) 1983-09-13 US disclosed
EP-0049728-A2 Method for enhancing the growth rate of meat-producing animals and for improving the lean meat to fat ratio thereof AMERICAN CYANAMID COMPANY (US) 1982-04-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250026721-A1 COMPOUNDS AND METHODS FOR MODULATING RAS-PI3K KRAS, HRAS, NRAS PRKCI 244/4885CREBBP 410/4885CA2 3649/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.