SCHEMBL8423136

SCHEMBL8423136

CCOC(=O)c1cccc(-c2cc(-c3ccc(Cl)cc3)nn2-c2ccc(S(N)(=O)=O)cc2)c1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 10/20 0.68
PTGS2 P35354 4/20 0.65
PTGS1 P23219 1/20 0.60
CA9 Q16790 3/20 0.59
CYP2C9 P11712 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA4 P22748 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420932 0.92 PTGS2 (0.59) CHRNA7PTGS2PTGS1CA9CYP2C9
SCHEMBL8119795 0.91 CHRNA7 (0.75) CHRNA7PTGS2PTGS1CA9SMN1; SMN2
SCHEMBL9253143 0.90 PTGS2 (0.66) CHRNA7PTGS2PTGS1CA9CYP2C9
SCHEMBL8126446 0.87 SMN1; SMN2 (0.70) CHRNA7PTGS2PTGS1CA9CYP2C9
SCHEMBL8120201 0.86 PTGS2 (0.66) CHRNA7PTGS2PTGS1CYP2C9SMN1; SMN2
SCHEMBL8119257 0.83 PTGS2 (0.67) CHRNA7PTGS2PTGS1CYP2C9SMN1; SMN2
SCHEMBL8119016 0.83 PTGS2 (0.72) CHRNA7PTGS2PTGS1CYP2C9SMN1; SMN2
SCHEMBL8423687 0.82 PTGS2 (0.66) CHRNA7PTGS2PTGS1CA9SMN1; SMN2
SCHEMBL8422291 0.81 PTGS2 (0.62) PTGS2PTGS1CA9SMN1; SMN2CA1
SCHEMBL8118945 0.81 PTGS2 (0.73) CHRNA7PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed