SCHEMBL8423752

SCHEMBL8423752

Cc1cccc(-c2cc(-c3ccc(Cl)cc3)nn2-c2ccccc2S(N)(=O)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.49
PTGS2 P35354 8/20 0.48
PTGS1 P23219 2/20 0.46
EGFR P00533 2/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CHRNA7 P36544 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CACNB4 O00305 2/20 0.38
CACNA1A O00555 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8422283 0.96 CYP2C9 (0.49) CYP2C9PTGS2PTGS1EGFRNPC1
SCHEMBL6903209 0.90 CYP2C9 (0.61) CYP2C9PTGS2PTGS1EGFRNPC1
SCHEMBL8424076 0.90 CYP2C9 (0.57) CYP2C9PTGS2PTGS1EGFRNPC1
SCHEMBL8422270 0.90 PTGS2 (0.48) CYP2C9PTGS2PTGS1NPC1RAB9A
SCHEMBL8422298 0.90 CYP2C9 (0.57) CYP2C9PTGS2PTGS1EGFRNPC1
SCHEMBL8421509 0.89 PTGS2 (0.50) CYP2C9PTGS2PTGS1CHRNA7CACNB4
SCHEMBL8733829 0.89 PTGS2 (0.54) CYP2C9PTGS2PTGS1EGFRNPC1
SCHEMBL8421778 0.89 PTGS2 (0.56) CYP2C9PTGS2PTGS1NPC1RAB9A
SCHEMBL8424034 0.88 PTGS2 (0.47) CYP2C9PTGS2PTGS1NPC1RAB9A
SCHEMBL8424132 0.88 PTGS2 (0.49) CYP2C9PTGS2PTGS1EGFRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed