SCHEMBL8733829

SCHEMBL8733829

NS(=O)(=O)c1ccccc1-n1nc(-c2ccccc2)cc1-c1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.54
CYP2C9 P11712 1/20 0.52
PTGS1 P23219 3/20 0.51
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MMP2 P08253 1/20 0.44
EGFR P00533 1/20 0.44
MAPK9 P45984 1/20 0.43
MARS1 P56192 1/20 0.43
AURKA O14965 1/20 0.42
APP P05067 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
PDPK1 O15530 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421778 0.97 PTGS2 (0.56) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL6903209 0.94 CYP2C9 (0.61) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL8422286 0.93 PTGS2 (0.52) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL8423767 0.93 PTGS2 (0.52) PTGS2CYP2C9PTGS1KDM4EMEN1
Methane SCHEMBL6309760 0.92 PTGS2 (0.47) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL8422373 0.92 CYP2C9 (0.55) PTGS2CYP2C9PTGS1MMP2EGFR
SCHEMBL8424076 0.92 CYP2C9 (0.57) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL8420732 0.92 PTGS2 (0.51) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL8423901 0.92 PTGS2 (0.51) PTGS2CYP2C9PTGS1KDM4EMEN1
SCHEMBL8423819 0.92 PTGS2 (0.51) PTGS2CYP2C9PTGS1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed