SCHEMBL8423800

SCHEMBL8423800

CS(=O)(=O)c1ccc(-n2nc(-c3ccc(Cl)cc3)cc2-c2cccc(O)c2)cc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.69
RARA P10276 4/20 0.59
RARB P10826 4/20 0.59
RARG P13631 4/20 0.59
RXRA P19793 4/20 0.59
PTGS1 P23219 2/20 0.54
ALOX5 P09917 1/20 0.50
CYP2C9 P11712 1/20 0.50
MMP2 P08253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8424552 0.96 PTGS2 (0.69) PTGS2RARARARBRARGRXRA
SCHEMBL8423820 0.90 PTGS2 (0.73) PTGS2RARARARBRARGRXRA
SCHEMBL8111976 0.89 PTGS2 (0.69) PTGS2PTGS1CYP2C9MMP2
SCHEMBL8420755 0.89 PTGS2 (0.79) PTGS2RARARARBRARGRXRA
SCHEMBL8423360 0.89 PTGS2 (0.79) PTGS2RARARARBRARGRXRA
SCHEMBL8420945 0.88 PTGS2 (0.71) PTGS2RARARARBRARGRXRA
SCHEMBL8421185 0.88 PTGS2 (0.80) PTGS2RARARARBRARGRXRA
SCHEMBL8420828 0.88 PTGS2 (0.80) PTGS2RARARARBRARGRXRA
SCHEMBL8420804 0.87 PTGS2 (0.88) PTGS2RARARARBRARGRXRA
SCHEMBL8423279 0.87 PTGS2 (0.72) PTGS2RARARARBRARGRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed
US-5434178-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G.D. SEARLE & CO. (US) 1995-07-18 US disclosed