SCHEMBL8423841

SCHEMBL8423841

COc1ccc(-c2cc(-c3ccc(Cl)cc3)n(-c3ccccc3S(N)(=O)=O)n2)cc1OC

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.68
PTGS1 P23219 1/20 0.52
CACNA1B Q00975 11/20 0.46
CACNB4 O00305 6/20 0.46
CACNA1A O00555 6/20 0.46
CACNA1G O43497 6/20 0.46
CACNG3 O60359 6/20 0.46
CACNA1F O60840 6/20 0.46
CACNA1H O95180 6/20 0.46
CACNB3 P54284 6/20 0.46
CACNA2D1 P54289 6/20 0.46
CACNG7 P62955 6/20 0.46
CACNA1D Q01668 6/20 0.46
CACNB1 Q02641 6/20 0.46
CACNG1 Q06432 6/20 0.46
CACNB2 Q08289 6/20 0.46
CACNA1S Q13698 6/20 0.46
CACNA1C Q13936 6/20 0.46
CACNA1E Q15878 6/20 0.46
CACNA2D4 Q7Z3S7 6/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421931 0.96 PTGS2 (0.63) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL8420715 0.88 PTGS2 (0.67) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL8421778 0.87 PTGS2 (0.56) PTGS2PTGS1MEN1MAPTKMT2A
SCHEMBL8421854 0.86 PTGS2 (0.50) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL8421630 0.86 PTGS2 (0.50) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL8733829 0.85 PTGS2 (0.54) PTGS2PTGS1MEN1KMT2ASMN1; SMN2
SCHEMBL8420748 0.84 PTGS2 (0.53) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL8421552 0.84 PTGS2 (0.53) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL7054592 0.84 PTGS2 (0.63) PTGS2PTGS1CACNA1BCACNB4CACNA1A
SCHEMBL8420838 0.84 PTGS2 (0.48) PTGS2PTGS1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed