SCHEMBL8423982

SCHEMBL8423982

N#Cc1ccc(-c2cc(-c3ccc(C#N)cc3)n(-c3ccccc3S(N)(=O)=O)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 3/20 0.46
CYP2C9 P11712 1/20 0.46
PTGES2 Q9H7Z7 1/20 0.42
CA12 O43570 1/20 0.40
CACNA1B Q00975 2/20 0.40
KDM1A O60341 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CACNB4 O00305 1/20 0.39
CACNA1A O00555 1/20 0.39
CACNA1G O43497 1/20 0.39
CACNG3 O60359 1/20 0.39
CACNA1F O60840 1/20 0.39
CACNA1H O95180 1/20 0.39
CACNB3 P54284 1/20 0.39
CACNA2D1 P54289 1/20 0.39
CACNG7 P62955 1/20 0.39
CACNA1D Q01668 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8422143 0.94 PTGS2 (0.48) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8423923 0.94 PTGS2 (0.48) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8422373 0.86 CYP2C9 (0.55) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8423066 0.86 MEN1 (0.45) PTGS2CYP2C9PTGES2MMP2
SCHEMBL8423874 0.85 CYP2C9 (0.49) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8423857 0.85 MEN1 (0.44) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8693648 0.84 PTGS2 (0.67) PTGS2CA1CA2CA9PTGES2
SCHEMBL8637681 0.84 PDPK1 (0.54) PTGS2CA1CA2CA9CYP2C9
SCHEMBL8421778 0.84 PTGS2 (0.56) PTGS2CYP2C9
SCHEMBL8421860 0.84 CYP2C9 (0.48) PTGS2CA1CA2CA9CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed