SCHEMBL8424022

SCHEMBL8424022

CC1=NN(c2ccccn2)C(=O)C1.CCOC(=O)CC(C)=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 10/20 0.67
PDCD1 Q15116 8/20 0.67
ALDH1A1 P00352 5/20 0.46
ATM Q13315 1/20 0.46
GAA P10253 2/20 0.42
MAPT P10636 4/20 0.42
KDM4E B2RXH2 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CHRM2 P08172 1/20 0.42
CYP3A4 P08684 1/20 0.42
CHRM1 P11229 1/20 0.42
TSHR P16473 1/20 0.42
PTGS1 P23219 1/20 0.42
DRD3 P35462 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3886681 0.82 CD274 (1.00) CD274PDCD1ALDH1A1GAAMAPT
SCHEMBL8425478 0.78 CD274 (0.48) CD274PDCD1ALDH1A1ATMGAA
SCHEMBL8425824 0.78 KMT2A (0.49) ALDH1A1GAAMAPTKDM4ESMN1; SMN2
SCHEMBL8427533 0.77 MAPT (0.65) ALDH1A1GAAMAPTKDM4ESMN1; SMN2
SCHEMBL8425552 0.76 POLB (0.55) ALDH1A1GAAMAPTKDM4ESMN1; SMN2
SCHEMBL8428070 0.74 CA1 (0.54) ALDH1A1GAAMAPTKDM4ESMN1; SMN2
SCHEMBL8425596 0.74 GAA (0.47) CD274PDCD1ALDH1A1GAAMAPT
SCHEMBL8428126 0.72 ALDH1A1 (0.43) ALDH1A1GAAMAPTKDM4ESMN1; SMN2
SCHEMBL8423248 0.72 APP (0.43) ALDH1A1GAAMAPTKDM4ESMN1; SMN2
SCHEMBL28847231 0.70 GAA (0.48) ALDH1A1ATMGAAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869516-A 4-(arylaminomethylene)-2,4-dihydro-3-pyrazolones MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-02-09 US disclosed