SCHEMBL8424062

SCHEMBL8424062

CN(C)C=Nc1ccc(Cl)cc1C#N

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
MAPT P10636 3/20 0.41
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NOS3 P29474 4/20 0.37
NOS1 P29475 4/20 0.37
NOS2 P35228 4/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
CYP2A6 P11509 1/20 0.35
VCAM1 P19320 1/20 0.35
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HPGD P15428 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29986270 1.00 GAA (0.42) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL4014542 0.83 GAA (0.44) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL4014545 0.83 GAA (0.44) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL14191690 0.83 GAA (0.44) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL14191688 0.82 CYP3A4 (0.49) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL1576898 0.81 GAA (0.45) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL1192238 0.81 ALDH1A1 (0.44) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL1822157 0.81 LMNA (0.42) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL1192235 0.81 ALDH1A1 (0.44) GAAMAPTKMT2AALDH1A1SMN1; SMN2
SCHEMBL5491257 0.81 LMNA (0.42) GAAMAPTKMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946549-A1 COMBINATORIAL PROCESS FOR PREPARING FUSED PYRIMIDINE LIBRARIES ELI LILLY AND COMPANY (US) 1999-10-06 EP disclosed
WO-1998027087-A1 COMBINATORIAL PROCESS FOR PREPARING FUSED PYRIMIDINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-06-25 WO disclosed