SCHEMBL8425432

SCHEMBL8425432

N#Cc1cccc(CN2CC(OS(=O)(=O)c3ccc4oc5ccccc5c4c3C(N)=O)CC2=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
ADRA1D P25100 1/20 0.34
JAK2 O60674 2/20 0.33
JAK1 P23458 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTR2B P41595 1/20 0.33
ALDH1A1 P00352 4/20 0.32
GLA P06280 1/20 0.32
JAK3 P52333 1/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
PDE10A Q9Y233 2/20 0.32
CFD P00746 1/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32
NPC1 O15118 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8423834 0.70 F10 (0.41) SIRT2SIRT1ADRA1DJAK2JAK1
SCHEMBL2333283 0.70 F10 (0.50) SIRT2SIRT1L3MBTL1ALDH1A1HPGD
SCHEMBL7415513 0.65 SIRT2 (0.51) SIRT2SIRT1ADRA1DL3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL2332921 0.65 SIRT2 (0.50) SIRT2SIRT1ADRA1DL3MBTL1ALDH1A1
SCHEMBL2330939 0.62 RORC (0.46) SIRT2SIRT1L3MBTL1ALDH1A1
SCHEMBL2325323 0.62 F10 (0.50) F10
SCHEMBL7427081 0.62 SIRT2 (0.60) SIRT2SIRT1ADRA1DL3MBTL1ROCK2
SCHEMBL6157745 0.61 HCRTR1 (0.48) HPGD
SCHEMBL2560664 0.59 PDE10A (0.70) L3MBTL1ALDH1A1PDE10AKDM4EHPGD
SCHEMBL7427087 0.59 SIRT2 (0.53) SIRT2SIRT1ADRA1DL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958918-A Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N- (aminominomethyl)phenylalkyl!-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. 1999-09-28 US disclosed