SCHEMBL8426327

SCHEMBL8426327

COc1cc(C(F)(F)F)cc(C(=O)NC(=N)N)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
GPR35 Q9HC97 2/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TMPRSS4 Q9NRS4 2/20 0.37
SCN8A Q9UQD0 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
CFTR P13569 1/20 0.35
NR2E1 Q9Y466 1/20 0.35
P2RX1 P51575 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8340423 0.99 MAPT (0.40) MAPTGPR35CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL8116539 0.85 CYP2C19 (0.40) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8428550 0.84 GPR35 (0.38) GPR35TMPRSS4P2RX1MEN1ALDH1A1
Hydrochloric Acid SCHEMBL8333007 0.83 GPR35 (0.37) GPR35TMPRSS4P2RX1MEN1ALDH1A1
SCHEMBL8116932 0.82 MAPT (0.47) MAPTSCN8ASCN10ACFTRKDM4E
SCHEMBL8428562 0.81 GPR35 (0.35) GPR35TMPRSS4P2RX1MEN1KMT2A
Hydrochloric Acid SCHEMBL8102752 0.81 MAPT (0.46) MAPTSCN8ASCN10ACFTRPPARA
SCHEMBL8430498 0.80 GPR35 (0.36) GPR35TMPRSS4P2RX1MEN1KMT2A
Hydrochloric Acid SCHEMBL8336174 0.80 GPR35 (0.35) GPR35TMPRSS4P2RX1MEN1KMT2A
SCHEMBL8428603 0.80 GPR35 (0.37) GPR35TMPRSS4P2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0791577-B1 Ortho-substituted benzylguanidines, process for their preparation and their use as medicament or diagnostic agent as well as medicament containing them HOECHST AG (DE) 1999-11-03 EP claimed