SCHEMBL8426437

SCHEMBL8426437

CC(C)(C)c1ccc(C(=O)NC(N)=NCl)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.38
NPFFR2 Q9Y5X5 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PLA2G1B P04054 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX12 P18054 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
NOTUM Q6P988 1/20 0.36
DDR1 Q08345 2/20 0.36
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
TAS1R2 Q8TE23 2/20 0.36
HDAC1 Q13547 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC3 O15379 1/20 0.35
RAF1 P04049 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8332845 0.99 PLAU (0.37) PLAUNPFFR2CYP1A2CYP2C19NPSR1
SCHEMBL8428730 0.85 NPSR1 (0.44) NPFFR2CYP1A2CYP2C19NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL8430572 0.84 NPSR1 (0.44) NPFFR2CYP1A2CYP2C19NPSR1ALDH1A1
SCHEMBL7797863 0.84 P4HB (0.38) NPFFR2CYP1A2CYP2C19NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL7791921 0.83 P4HB (0.38) NPFFR2CYP1A2CYP2C19NPSR1ALDH1A1
SCHEMBL8428715 0.82 SIRT1 (0.46) CYP1A2CYP2C19NPSR1ALDH1A1CYP2C9
SCHEMBL8428392 0.82 SCN5A (0.42) NPFFR2CYP1A2CYP2C19NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL8426168 0.81 SIRT1 (0.46) CYP1A2CYP2C19NPSR1ALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL8333476 0.81 SCN5A (0.41) NPFFR2CYP1A2CYP2C19NPSR1ALDH1A1
Hydrochloric Acid SCHEMBL8655513 0.79 TOP1 (0.39) NPFFR2CYP2C19ALDH1A1CYP2C9HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0791577-B1 Ortho-substituted benzylguanidines, process for their preparation and their use as medicament or diagnostic agent as well as medicament containing them HOECHST AG (DE) 1999-11-03 EP claimed