SCHEMBL8426656

SCHEMBL8426656

N#CCC1CCc2ccccc2O1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.51
HTR1A P08908 12/20 0.49
SIGMAR1 Q99720 2/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
HTR1D P28221 10/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29698783 1.00 CA2 (0.51) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL8425962 0.84 CA2 (0.49) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL2325413 0.83 CA2 (0.55) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL8089401 0.83 HRH3 (0.46) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL4936360 0.79 CA2 (0.56) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL4936349 0.79 CA2 (0.56) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL8049371 0.78 HTR1A (0.60) CA2HTR1AHTR1D
SCHEMBL8640922 0.78 CA2 (0.47) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL8879867 0.78 HTR1A (0.60) CA2HTR1AHTR1D
SCHEMBL6348788 0.77 HTR1A (0.56) CA2HTR1ASIGMAR1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925662-A OXIDASE INHIBITORS SYNTHELABO (FR) 1999-07-20 US disclosed
US-5112855-A Nootropic Agents CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
US-4957928-A NOOTROPIC AGENTS, COGNITION ACTIVATORS CIBA-GEIGY CORPORATION (US) 1990-09-18 US disclosed
EP-0252005-A1 Hydrogenated 1-benzooxacycloalkyl-pyridine carboxylic-acid compounds CIBA-GEIGY AG (CH) 1988-01-07 EP disclosed