SCHEMBL8426685

SCHEMBL8426685

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(N)s1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.53
CTSS P25774 5/20 0.47
CTSK P43235 4/20 0.47
ITGB3 P05106 2/20 0.47
ITGA2B P08514 2/20 0.47
PTPN1 P18031 1/20 0.46
PPARA Q07869 6/20 0.46
PPARG P37231 5/20 0.46
SCN9A Q15858 1/20 0.45
ITGB1 P05556 1/20 0.45
ITGAV P06756 1/20 0.45
ITGB5 P18084 1/20 0.45
PPARD Q03181 2/20 0.44
ITGA4 P13612 1/20 0.44
ITGB7 P26010 1/20 0.44
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8426686 1.00 ACE (0.53) ACECTSSCTSKITGB3ITGA2B
SCHEMBL8530056 0.90 CTSS (0.45) ACECTSSCTSKCTSLCTSB
SCHEMBL8530060 0.90 CTSS (0.45) ACECTSSCTSKCTSLCTSB
SCHEMBL8426689 0.86 ALDH1A1 (0.48) ACECTSSCTSKSCN9ACTSL
SCHEMBL8426691 0.86 ALDH1A1 (0.48) ACECTSSCTSKSCN9ACTSL
SCHEMBL25177899 0.85 ACE (0.50) ACECTSSCTSKITGB3ITGA2B
SCHEMBL539422 0.85 ACE (0.50) ACECTSSCTSKITGB3ITGA2B
SCHEMBL3376657 0.85 ACE (0.50) ACECTSSCTSKITGB3ITGA2B
SCHEMBL8526061 0.81 ACE (0.45) ACECTSSCTSKITGB3ITGA2B
SCHEMBL8526064 0.81 ACE (0.45) ACECTSSCTSKITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874472-A Aminoacid derivatives as no synthase inhibitors GLAXO WELLCOME INC. (US) 1999-02-23 US disclosed
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed