SCHEMBL8427008

SCHEMBL8427008

Clc1ccc(/C=C/C2=CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
KMT2A Q03164 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
MEN1 O00255 1/20 0.50
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
BCHE P06276 2/20 0.46
ACHE P22303 2/20 0.46
BACE1 P56817 2/20 0.46
OPRM1 P35372 1/20 0.45
OPRK1 P41145 1/20 0.45
DRD4 P21917 3/20 0.44
DRD3 P35462 2/20 0.44
DRD2 P14416 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8427010 1.00 KDM4E (0.62) KDM4ESMN1; SMN2KMT2ASIGMAR1MEN1
SCHEMBL8429502 0.95 KDM4E (0.62) KDM4ESMN1; SMN2KMT2ASIGMAR1MEN1
SCHEMBL8429499 0.95 KDM4E (0.62) KDM4ESMN1; SMN2KMT2ASIGMAR1MEN1
SCHEMBL8426856 0.93 KDM4E (0.70) KDM4ESMN1; SMN2DRD4DRD3DRD2
SCHEMBL8426855 0.93 KDM4E (0.70) KDM4ESMN1; SMN2DRD4DRD3DRD2
SCHEMBL8429501 0.92 KDM4E (0.64) KDM4ESMN1; SMN2KMT2ASIGMAR1NPC1
SCHEMBL8429503 0.92 KDM4E (0.64) KDM4ESMN1; SMN2KMT2ASIGMAR1NPC1
Hydrochloric Acid SCHEMBL8428835 0.90 KDM4E (0.66) KDM4ESMN1; SMN2KMT2ANPC1RAB9A
Hydrochloric Acid SCHEMBL8428831 0.90 KDM4E (0.66) KDM4ESMN1; SMN2KMT2ANPC1RAB9A
SCHEMBL8128377 0.88 SMN1; SMN2 (0.60) KDM4ESMN1; SMN2KMT2ASIGMAR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861407-A Tetrahydropyridine derivatives as dopamine receptor subtype ligands MERCK SHARP & DOHME, LTD. (GB) 1999-01-19 US disclosed