SCHEMBL8428388

SCHEMBL8428388

CC(C)c1cc(Cl)c(C(=O)NC(=N)N)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.39
CTSS P25774 2/20 0.37
CTSK P43235 1/20 0.37
KDM4E B2RXH2 3/20 0.35
MAPT P10636 2/20 0.34
TP53 P04637 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 1/20 0.34
APEX1 P27695 1/20 0.34
ALDH1A1 P00352 3/20 0.33
GAA P10253 3/20 0.33
TRPA1 O75762 2/20 0.32
PDE2A O00408 1/20 0.32
PDK1 Q15118 1/20 0.32
F7 P08709 1/20 0.31
KDR P35968 1/20 0.31
ALOX12 P18054 1/20 0.31
TMPRSS4 Q9NRS4 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8333467 0.99 S1PR1 (0.38) S1PR1CTSSCTSKKDM4EMAPT
SCHEMBL8428726 0.83 TP53 (0.39) CTSSCTSKKDM4EMAPTTP53
SCHEMBL8426433 0.82 POLB (0.38) CTSSCTSKKDM4EMAPTTP53
Hydrochloric Acid SCHEMBL8337102 0.82 TP53 (0.38) CTSSCTSKKDM4EMAPTTP53
SCHEMBL7797854 0.81 TMPRSS4 (0.41) KDM4EMAPTTP53RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL8332842 0.81 POLB (0.38) CTSSCTSKKDM4EMAPTTP53
Hydrochloric Acid SCHEMBL7791912 0.80 TMPRSS4 (0.40) KDM4EMAPTTP53RAB9ASMN1; SMN2
SCHEMBL8428710 0.80 MAPT (0.40) S1PR1MAPTRAB9AGAAMEN1
Hydrochloric Acid SCHEMBL8335173 0.79 MAPT (0.40) S1PR1MAPTRAB9AGAAMEN1
SCHEMBL8430503 0.78 SMN1; SMN2 (0.33) S1PR1MAPTTP53RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0791577-B1 Ortho-substituted benzylguanidines, process for their preparation and their use as medicament or diagnostic agent as well as medicament containing them HOECHST AG (DE) 1999-11-03 EP claimed